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| Item No | Product Name | Product Description | Product Description | Inquiry |
|---|---|---|---|---|
| R-SX-407 | Ambrisentan; BSF208075; LU208075,CAS177036-94-1 | Ambrisentan 是一種選擇性的ET A型受體 (ETAR) 拮抗劑。 西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
| R-SX-408 | Empagliflozin，CAS864070-44-0 | Empagliflozin是一種選擇性鈉葡萄糖協(xié)同轉(zhuǎn)運(yùn)蛋白-2 (SGLT-2) 抑制劑，抑制人SGLT-2的IC50 為3.1 nM。西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
| R-SX-409 | Canagliflozin hemihydrate,CAS928672-86-0 | Canagliflozin 0.5 H2O(JNJ 28431754; TA 7284) is a highly potent and selective SGLT2 inhibitor for hSGLT2 with IC50 of 2.2 nM, exhibits 413-fold selectivity over hSGLT1. IC50 value: 2.2 Nm西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
| R-SX-410 | Ipragliflozin,CAS761423-87-4 | Ipragliflozin (ASP1941) is a highly potent and selective SGLT2 inhibitor with IC50 of 2.8 nM; little and NO potency for SGLT1/3/4/5/6. IC50 value: 2.8 nM.西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
| R-SX-411 | Tofogliflozin,CAS1201913-82-7 | Tofogliflozin(CSG-452) hydrate is a potent and highly specific sodium/glucose cotransporter 2(SGLT2) inhibitor with Ki values of 2.9, 14.9, and 6.4 nM for human, rat, and mouse SGLT2. IC50 value: 2.9/14.9/6.4 nM(human/rat/mouse SGLT2)西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
| R-SX-412 | Plerixafor; AMD310,CAS110078-46-1 | Plerixafor (AMD3100) is a chemokine receptor antagonist for CXCR4 and CXCL12-mediated chemotaxis with IC50 of 44 nM and 5.7 nM in cell-free assays, respectively.西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
| R-SX-413 | Reversine,CAS656820-32-5 | Reversine 是一種ATP-競(jìng)爭(zhēng)性的 Aurora kinase 抑制劑，作用于 Aurora A，Aurora B 和 Aurora C，IC50 分別為 400，500 和 400 nM。西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
| R-SX-414 | CYM5442,CAS1094042-01-9 | CYM 5442 HCl is a potent and selective EDG-1 (S1P1) agonist in vitro (EC50 = 1.35 nM).西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
| R-SX-415 | Capadenoson; BAY 68-4986,CAS544417-40-5 | Capadenoson (BAY 68-4986) is a new adenosine A1 receptor agonist.西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
| R-SX-416 | Ki16198,CAS355025-13-7 | Ki16198 is the methyl ester of Ki16425, which is a LPA antagonist and inhibits LPA1- and LPA3-induced inositol phosphate production with Ki of 0.34 μM and 0.93 μM, respectively, shows weaker inhibition for LPA2, no activity at LPA4, LPA5, LPA6.西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
| R-SX-417 | ozanimod;RPC1063;RPC-1063,CAS1306760-87-1 | Ozanimod 是一種有效的選擇性 S1P1 和 S1P5 受體激動(dòng)劑，在[35S]-GTPγS 結(jié)合實(shí)驗(yàn)中，EC50 分別為 410±160 pM 和 11±4.3 nM。西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
| R-SX-418 | ABC294640,CAS915385-81-8 | ABC294640 is an orally bioavailable and selective sphingosine kinase-2 (SphK2) inhibitor with IC50 of approximately 60 μM. Phase 1/2.西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
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